at Peking University School of Pharmaceutical Sciences
中文版
​​​​the Jia Research Group
Independent research
111. “Total Synthesis of (+)-Kalmanol”, Tianhao Ma, Yiming Ma, Bo Li, Yanxing Jia*. Angew. Chem. Int. Ed. 2024, e202407215.
Download →
110. “Twenty-Step Total Synthesis of (+)-Phorbol”, Kuan Zhao, Yifu Cheng, Yanxing Jia*. CCS Chem. 2024, Just Published. DOI: 10.31635/ccschem.024.202404505.
Download →
109. “Biomimetic synthesis of pallavicinin, neopallavicinin, pallambins A–D, pallaviambins A/B, and pallavicinolides B/C”, Lijun Chen, Peng Chen, Xiwu Zhang, Yu Zhang, Yanxing Jia*. Chem 2024, https://doi.org/10.1016/j.chempr.2024.04.003.
Download →
108. “Gut symbionts alleviate MASH through a secondary bile acid biosynthetic pathway”, Qixing Nie, Xi Luo, Kai Wang, Yong Ding, Shumi Jia, Qixiang Zhao, Meng Li, Jinxin Zhang, Yingying Zhuo, Jun Lin, Chenghao Guo, Zhiwei Zhang, Huiying Liu, Guangyi Zeng, Jie You, Lulu Sun, Hua Lu, Ming Ma,  Yanxing Jia*, Ming-Hua Zheng*, Yanli Pang*, Jie Qiao*, Changtao Jiang*. Cell 2024, https://doi.org/10.1016/j.cell.2024.03.034.
Download →
107. “Total Synthesis of Pallamolides A−E”, Yu Zhang, Lijun Chen, Yanxing Jia*. Angew. Chem. Int. Ed. 2024, e202319127.
Download →
106. “Bioinspired Total Syntheses of Grayanotoxins II/III, Kalmanol, and Rhodomollacetals A–C with Three Distinct Skeletons”, Hao Cheng, Tianhao Ma, Xiao Liu, Yanxing Jia*. CCS Chem. 2024, Just Published. DOI: 10.31635/ccschem.024.202303731.
Download →
105. “Bioinspired Total Synthesis of Bipolarolides A and B”, Bo Li, Chuanzhen Tan, Tianhao Ma, Yanxing Jia*. Angew. Chem. Int. Ed. 2024, e202319306.
Download →
104. “Design, syntheses and biological evaluation of natural product aiphanol derivatives and analogues: Discovery of potent anticancer agents”, Licheng Yao, Wenqing Cai, Shanmei Chen, Aidan Wang, Xin Wang, Chuanke Zhao, Chengchao Shou*, Yanxing Jia*. Bioorg. Med. Chem. Lett. 2023, 90, 129326.
Download →

103. “Total Synthesis of (+)-Aberrarone”, Yang Wang, Yongjian Su, Yanxing Jia*. J. Am. Chem. Soc. 2023, 145, 9459-9463.

          Organic Chemistry Portal (https://www.organic-chemistry.org/Highlights/2023/06November.shtm), D. F. Taber.

Download →
102. “Total Synthesis of (−)-Principinol C”, 
  • Tianhao Ma
    • , 
  • Hao Cheng
    • , 
  • Mallesham Pitchakuntla
    • , 
  • Weihao Ma
    • , Yanxing Jia*. J. Am. Chem. Soc. 2022, 144, 20196-20200.
    Download →
    Download →

    100. “Bioinspired Total Synthesis of (+)-Euphorikanin A”, Zhuang Chen, Kuan Zhao, Yanxing Jia*. Angew. Chem. Int. Ed. 2022, 61, e202200576.

    Download →
    Download →
    99. “Cascade Cyclization Reaction Initiated by Benzylic Carbocation of Indole: Scope and Mechanistic Insights”, Zhongrun Gao, Yuan Wang, Hang Song, Zhengren Xu*, Yanxing Jia*. Chin. J. Org. Chem. 2021, 41, 3126-3133.
    Download →
    98. “Protecting-Group-Free Total Synthesis of (–)-Pallambins A-D”, Xiwu Zhang, Yuan Wang, Peng Chen, Xinxian Cai, Yanxing Jia*. Chin. J. Chem. 2021, 39, 1983-1996.
    Download →
    97. “Total synthesis of Kopsine, Fruticosine, and structurally related polycyclic caged Kopsia indole alkaloids”, Bo Qin, Yuan Wang, Xin Wang*, Yanxing Jia*. Org. Chem. Front. 2021, 8(2), 3​69-383.
    96. “Synthesis of benzofuro[3,2-b]indolines via regioselective electrooxidative coupling of indoles and phenols”, Keyuan Li, Yuan Wang, Lijun Chen, Lei Li, Yanxing Jia*. Tetrahedron. Lett. 2021, 63(36), 152603.
    Download →
    95. “Total Synthesis of (−)-Glaucocalyxin A”, Jiuzhou Guo, Bo Li, Weihao Ma, Mallesham Pitchakuntla, Yanxing Jia*. Angew. Chem. Int. Ed. 2020, 59(35), 15195–15198. Angew. Chem. 2020, 132(35), 15307–15310.

    highlighted in synfacts, Synfacts 2020, 16(08), 0882.

    《有机化学》亮点介绍，2020, 40(10), 3487-3489.

    Download →
    94. “Seven-step total synthesis of α-cyclopiazonic acid”, Shibin Shi, Kuo Yuan, Yanxing Jia*. Chin. Chem. Lett. 2020, 31(2), 401–403.
    Download →
    93. “A concise total synthesis of secoisolariciresinol”, Jiuzhou Guo, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(10), 699–703.
    Download →
    92. “Improved synthesis of key intermediate of grayanotoxin III”, Weihao Ma, Zhi Huang, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(6), 402–407.
    Download →
    91. “Type-II Pauson-Khand Reaction of 1,8-enyne in the Attempt of Building 7/5 Ring of (-)-Caribenol A and DFT Understanding”, Yang Wang, Kang Liu, Zhi-Xiang Yu*, Yanxing Jia*. Tetrahedron Lett. 2019, 60(36), 151001 .
    Download →
    90. “Natural product incarvillateine aggravates epileptic seizures by inhibiting GABAA currents”, Xiling Bian*, Yu Zhang, Bin Huang, Xintong Wang, Gongxin Wang, Yuhao Zhu, Yan Liu, Jianhui Liang, Yanxing Jia*, Kewei Wang*. Eur. J. Pharmaco. 2019, 858, 172496.
    Download →
    89. “Enantioselective Total Syntheses of Pallambins A-D”, Xiwu Zhang, Xinxian Cai, Bin Huang, Lei Guo, Zhongrun Gao, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(38), 13380–13384. Angew. Chem. 2019, 131(38), 13514–13518.
    Download →
    88. “A Ten-Step Total Synthesis of Speradine C”, Haichao Liu, Lijun Chen, Kuo Yuan, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(19), 6362–6365. Angew. Chem. 2019, 131(19), 6428–6431.

    highlighted in synfacts, Synfacts 2019, 15(7), 0714.

         《有机化学》亮点介绍，2019, 39(8), 2344.

    Download →
    87. “Eight-Step Total Synthesis of Phalarine by Bioinspired Oxidative Coupling of Indole and Phenol”, Lei Li, Kuo Yuan, Qianlan Jia, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(18), 6074–6078. Angew. Chem. 2019, 131(18), 6135–6139.

    highlighted in synfacts, Synfacts 2019, 15(7), 0712.

    x-mol化学资讯平台亮点介绍.

    Download →
    86. “Synthetic approaches to natural products containing a 2,3-dihydrobenzofuran skeleton”, Zhuang Chen, Mallesham Pitchakuntla, Yanxing Jia*. Nat. Prod. Rep. 2019, 36(4), 666–690.
    Download →
    85. “Recent Progress in the Synthesis of 3,4-Fused Indole Alkaloids” “3,4-桥环吲哚类生物碱的合成进展”, Kuo Yuan, Yanxing Jia*. Chin. J. Org. Chem. 2018, 38(9), 2386-2399. 《有机化学》，2018, 38(9), 2386-2399.
    Download →
    84. “Divergent Strategy in Natural Product Total Synthesis”, Lei Li, Zhuang Chen, Xiwu Zhang, Yanxing Jia*. Chem. Rev. 2018, 118(7), 3752–3832.
    Download →
    83. “Synthetic Study toward the Total Synthesis of Fumigaclavines A–D”, Yongfan Ma, Yanxing Jia*. J. Chin. Pharm. Sci. 2017, 26(7), 496–503.
    Download →
    82. “Regioselective Direct C-4 Functionalization of Indole: Total Syntheses of (–)-Agroclavine and (–)-Elymoclavine”, Jianbo Lv, Bin Wang, Kuo Yuan, Yuan Wang, Yanxing Jia*. Org. Lett. 2017, 19(13), 3664– 3667.
    Download →
    81.“Total Syntheses of Festuclavine, Pyroclavine, Costaclavine, epi-Costaclavine, Pibocin A, 9-Deacetoxyfumigaclavine C, Fumigaclavine  G, and Dihydrosetoclavine”, Haichao Liu, Xiwu Zhang, Dong Shan, Mallesham Pitchakuntla, Yongfan Ma, Yanxing Jia*. Org. Lett. 2017, 19(12), 3323–3326.
    Download →
    80. “Total Syntheses of Naucleamides A−C and E, Geissoschizine, Geissoschizol, (E)-Isositsirikine, and 16-epi-(E)-Isositsirikine”, Lei Li, Paruke Aibibula, Qianlan Jia, Yanxing Jia*. Org. Lett. 2017, 19(10), 2642– 2645.
    Download →
    79.“Total synthesis of natural spiro-trisindole enantiomers similisines A, B and their stereoisomers”, Lunyong Shi, Lingyu Li, Jun Wang, Bin Huang, Kewu Zeng, Hongwei Jin, Qingying Zhang*, Yanxing Jia*. Tetrahedron Lett. 2017, 58(20), 1934–1938.
    Download →
    78. “Ergot alkaloids: synthetic approaches to lysergic acid and clavine alkaloids”, Haichao Liu, Yanxing Jia*. Nat. Prod. Rep. 2017, 34(4), 411–432.
    Download →
    77. “A Simple and Efficient Synthesis of Secondary Alkylamines from Nitroalkanes”, Zhi Huang, Jianbo Lu, Yanxing Jia*. ChemistrySelect. 2016, 1(18), 5892–5894.
    Download →
    76. “A concise gram-scale synthesis of ht-13-A via a rhodium-catalyzed intramolecular C–H activation reaction”, Pengyu Tao, Zhuang Chen, Yanxing Jia*. Chem. Commun. 2016, 52(75), 11300–11303.
    Download →
    75. “C–H bond activation in the total syntheses of natural products”, Pengyu Tao, Yanxing Jia*. Sci. China Chem. 2016, 59(9), 1109–1125.
    Download →
    74. “A palladium-catalyzed intramolecular carbonylative annulation reaction to form 4,5-fused tricyclic 2-quinolones”, Xiwu Zhang, Haichao Liu, Yanxing Jia*. Chem. Commun. 2016, 52(49), 7665–7667.

    highlighted in synfacts, Synfacts 2016, 12(9), 0896.

    Download →
    73. “Gram Scale Syntheses of (-)-Incarvillateine and Its Analogs. Discovery of Potent Analgesics for Neuropathic Pain”, Bin Huang, Fengying Zhang, Gang Yu, Yan Song, Xintong Wang, Meiliang Wang, Zehui Gong, Ruibin Su, Yanxing Jia*. J. Med. Chem. 2016, 59(8), 3953–3963 .
    Download →
    72. “Asymmetric Total Synthesis of 3-epi-naucleamide A”, Paruke Aibibula, Zhi Huang, Hong-Zheng Fu,* Yanxing Jia*. J. Chin. Pharm. Sci. 2016, 25(1), 30–36.
    Download →
    71. “Formal Synthesis of (+)-Kopsihainanine A and Synthetic Study toward (+)-Limaspermidine”, Zhuang Chen, Shiqiang Zhou, Yanxing Jia*. J. Org. Chem. 2015, 80(24), 12545–12551.
    Download →
    70. “Antinociceptive effects of incarvillateine, a monoterpene alkaloid from Incarvillea sinensis, and possible involvement of the adenosine system”, Mei-Liang Wang, Gang Yu*, Shou-Pu Yi, Feng-Ying Zhang, Zhi-Tong Wang, Bin Huang, Rui-Bin Su*, Yan-Xing Jia, Ze-Hui Gong. Sci. Rep. 2015, 5, 16107.
    Download →
    69. “Protecting-Group-Free Enantioselective Synthesis of (-)-Pallavicinin and (+)-Neopallavicinin”, Bin Huang, Lei Guo, Yanxing Jia*. Angew. Chem. Int. Ed. 2015, 54(46), 13599–13603. Angew. Chem. 2015, 127(46), 13803–13807.

    highlighted in synfacts, Synfacts 2015, 11(12), 1242.

    Organic Chemistry Portal (http://www.organic-chemistry.org/Highlights /2016/01August. shtm), D. F. Taber.

    x-mol化学资讯平台（http://www.x-mol.com/news/1398）亮点介绍 .

    Download →
    68. “Catalytic Asymmetric Total Synthesis of (-)-Galanthamine and (-)-Lycoramine”, Lei Li, Qiao Yang, Yuan Wang, Yanxing Jia*. Angew. Chem. Int. Ed. 2015, 54(21), 6255–6259. Angew. Chem. 2015, 127(21), 6353–6357.

    highlighted in synfacts, Synfacts 2015, 11(7), 0688.

    Organic Chemistry Portal（http://www.organic-chemistry.org/Highlights/2015 /30November.shtm）

    D. F. Taber, Org. Chem. Highlights 2015, November 30. Alkaloid Synthesis.

    《有机化学》亮点介绍，2015, 35(8), 1804.

    Download →
    67. “Asymmetric Total Synthesis of (+)–Dragmacidin D Reveals Unexpected Stereo Complexity”, Fengying Zhang, Bin Wang, Pritesh Prasad, Robert J. Capon, Yanxing Jia*. Org. Lett. 2015, 17(6), 1529–1532.
    Download →
    66. “Concise Synthesis of the Tricyclic Skeleton of Crotobarin and Crotogoudin via a Gold-catalyzed Cycloisomerization Reaction”, Yinliang Guo, Qiang Liu, Yanxing Jia*. Chem. Commun. 2015, 51(5), 889–891.
    Download →
    65. “Total Synthesis of (-)-Decursivine and Analogues via Cascade Sequence”, Fengying Zhang, Lei Li, Weimin Hu, Yanxing Jia*. Tetrahedron 2015, 71(22),  3756–3762. (Invited by Tetrahedron Symposium-in-Print (TSIP issue) focusing on “The Chemistry of Pyrrole and Indole Natural Products”, Edited by Ang Li)
    Download →
    64. “Synthetic studies of cyclic peptides stephanotic acid methyl ester, celogentin C and moroidin”, Lei Li, Weimin Hu, Yanxing Jia*. Tetrahedron 2014, 70(42),  7753–7762. (Invited by Tetrahedron Symposium-in-Print (TSIP issue) focusing on “Peptide macrocycles”, Edited by Lei Liu)
    Download →
    63. “Total Synthesis of Dictyodendrins B and E, and Formal Synthesis of Dictyodendrin C”, Pengyu Tao, Jingjing Liang, Yanxing Jia*. Eur. J. Org. Chem. 2014, 5735–5748.
    Download →
    62. “Total Synthesis of (-)-Goniomitine”, Shiqiang Zhou, Yanxing Jia*. Org. Lett. 2014, 16(12), 3416–3418.
    Download →
    61. “Rhodium-catalyzed intramolecular annulation via C-H activation leading to fused tricyclic indole scaffolds”, Pengyu Tao, Yanxing Jia*. Chem. Commun. 2014, 50(55), 7367–7370.
    Download →
    60. “Intramolecular Larock Indole Synthesis for the Preparation of Tricyclic Indoles and Its Application in the Synthesis of Tetrahydropyrroloquinoline and Fargesine”, Yan Gao, Dong Shan, Yanxing Jia*. Tetrahedron 2014, 70(34), 5136–5147. (Invited by Tetrahedron Symposium-in-Print (TSIP issue) focusing on “indole and pyrrole synthesis”)
    Download →
    59. “Palladium-catalyzed synthesis of benzofurans via C–H activation/oxidation tandem reaction and its application to the synthesis of decursivine and serotobenine”, Lei Guo, Fengying Zhang, Weimin Hu, Lei Li, Yanxing Jia*. Chem. Commun. 2014, 50(25), 3299–3302.
    Download →
    58. “Synthesis of the cycloheptannelated indole fragment of dragmacidin E”, Bin Wang, Hua Qin, Fengying Zhang, Yanxing Jia*. Tetrahedron Lett. 2014, 55(9), 1561–1563.
    Download →
    57. “Oxyfadichalcones A-C: three chalcone dimers fused through a cyclobutane ring from Tibetan medicine Oxytropis falcata Bunge”, Xiaojing Zhang, Lingyu Li, Shanshan Wang, Sheng Que, Wenzhi Yang, Fengying Zhang, Ningbo Gong, Wei Cheng, Hong Liang, Min Ye, Yanxing Jia, Qingying Zhang*. Tetrahedron 2013, 69(52), 11074–11079.
    Download →
    56. “Total Synthesis of (+)-Lysergic acid”, Qiang Liu, Yu-An Zhang, Ping Xu, Yanxing Jia*. J. Org. Chem. 2013, 78(21), 10885–10893.
    Download →
    55. “Direct Olefination at the C-4 Position of Tryptophan via C-H Activation: Application to Biomimetic Synthesis of Clavicipitic Acid”, Qiang liu, Qingjiang Li, Yongfan Ma, Yanxing Jia*. Org. Lett. 2013, 15(17), 4528–4531.
    Download →
    54. “Reagent-free synthesis of 2,3,4-polysubstituted tetrahydroquinolines: application to the formal synthesis of (±)-martinellic acid and martinelline”, Zhouting Rong, Qingjiang Li, Wenhan Lin*, Yanxing Jia*. Tetrahedron Lett. 2013, 54(33), 4432–4434.
    Download →
    53. “Construction of the A ring of halichomycin via a RCM strategy”, Shiyong Mao, Yanxing Jia*. Tetrahedron Lett. 2013, 54(32), 4343–4345 .
    Download →
    52. “Total Synthesis of Rugulovasine A”, Yu-An Zhang, Qiang liu, Chao Wang, Yanxing Jia*. Org. Lett. 2013, 15(14), 3662–3665.
    Download →
    51. “Total Synthesis of Dictyodendrin B and E”, Jingjing Liang, Weimin Hu, Pengyu Tao, Yanxing Jia*. J. Org. Chem. 2013, 78(11), 5810-5815.
    Download →
    50. “Progress in Synthesis of 3,4-Fused Indole Alkaloids” “3,4-桥环吲哚类生物碱的合成研究进展”, Dong Shan, Yanxing Jia*. Chin. J. Org. Chem. 2013, 33(6), 1144-1156. 《有机化学》，2013, 33(6), 1144-1156.（封面文章）
    Download →
    49. “Intramolecular Larock Indole Synthesis: Preparation of 3,4-Fused Tricyclic Indoles and Total Synthesis of Fargesine”, Dong Shan, Yan Gao, Yanxing Jia*. Angew. Chem. Int. Ed. 2013, 52(18), 4902–4905. Angew. Chem. 2013, 125(18), 5002–5005.

    (highlighted in synfacts, Synfacts 2013, 9(7), 0709)

    《有机化学》亮点介绍，2013, 33(8), 1334.

    Download →
    48. “Total Synthesis of (+)- and (-)-Decursivine and (±)-Serotobenine via a Cascade Witkop Photocyclization/Elimination/Addition Sequence: Scope and Mechanistic Insights”, Weimin Hu, Hua Qin, Yuxin Cui, Yanxing Jia*. Chem. Eur. J. 2013, 19(9), 3139–3147.
    Download →
    47. “Structural Optimization and Evaluation of Butenolides as Potent Antifouling Agents: Modification of the Side Chain Affects the Biological Activities of Compounds”, Yongxin Li, Fengying Zhang, Ying Xu, Kiyotaka Matsumura, Zhuang Han, Lingli Liu, Wenhan Lin, Yanxing Jia, Pei-Yuan Qian*. Biofouling 2012, 28(8), 857–864.
    Download →
    46. “Nine 2-(2-Phenylethyl)chromone Derivatives from the Resinous Wood of Aquilaria Sinensis and Their Inhibition of LPS-Induced NO Production in RAW 264.7 Cells”, Dong Chen, Zhengren Xu, Xingyun Chai, Kewu Zeng, Yanxing Jia, Dan Bi, Zhizhong Ma, Pengfei Tu*. Eur. J. Org. Chem. 2012, 5389–5397.
    Download →
    45. “Stereoselective Synthesis of the C5–C18 Fragment of Halichomycin”, Qingjiang Li, Shiyong Mao, Yuxin Cui, Yanxing Jia*. J. Org. Chem. 2012, 77(8), 4111–4116.
    Download →
    44. “Mg(ClO4)2-Catalyzed Intramolecular Allylic Amination: Application to the Total Synthesis of Demethoxyfumitremorgin C”, Danfeng Jiang, Zhengren Xu, Yanxing Jia*. Tetrahedron 2012, 68(22), 4225–4232.
    Download →
    43. “CuI-catalyst N-arylation of 4-Iodotryptophan Derivatives; Effort toward the Total Synthesis of Indolactam V”, Jingqiang Jiang, Zhengren Xu, Yanxing Jia*. J. Chin. Pharm. Sci. 2012, 21(2), 113–123.
    Download →
    42. “Total Synthesis of Maremycins A, B, C1/C2, D1, and D2”, Yonghua Liu, Liangren Zhang, Yanxing Jia*. Tetrahedron Lett. 2012, 53(6), 684–687.
    Download →
    41. “Total Synthesis of (+)-Lysergic acid”, Qiang Liu, Yanxing Jia*. Org. Lett. 2011, 13(18), 4810–4813.
    Download →
    40. “Recent Research Progress in the Research on Lamellarins and Related Pyrrole-derived Alkaloids from Marine Organisms”, Aili Fan, Wenhan Lin, Yanxing Jia*. J. Chin. Pharm. Sci. 2011, 20(5), 425–441. (Invited review)
    Download →
    39. “Domino Palladium-Catalyzed Heck/C-H Activation/Intermolecular Direct Arylation Reactions”, Zhiyao Lü, Yuxin Cui*, Yanxing Jia*. Synthesis 2011, 2595–2599. (Invited paper, a Special Topic on "C–H Functionalization/Activation" in SYNTHESIS)
    Download →
    38. “Total Synthesis of (±)-Decursivine and (±)-Serotobenine: A Witkop Photocyclization/Elimination/O-Michael Addition Cascade Approach”, Hua Qin, Zhengren Xu, Yuxin Cui, Yanxing Jia*. Angew. Chem. Int. Ed. 2011, 50(19), 4447–4449. Angew. Chem. 2011, 123(19), 4539–4541.

    (highlighted in synfacts, Synfacts 2011, 7(9), 0929-0929)

    D. F. Taber, Org. Chem. Highlights 2011, November 21. C-N Ring Construction: The Synthesis of Decursivine by Mascal and by Jia

         《有机化学》亮点介绍，2011, 31(8), 1334.

    Download →
    37. “Total Synthesis of (-)-Indolactam V”, Zhengren Xu, Fengying Zhang, Lihe Zhang, Yanxing Jia*. Org. Biomol. Chem. 2011, 9, 2512–2517.
    Download →
    36. “Total Synthesis of Lamellarins D, H, and R and Ningalin B”, Qingjiang Li, Jingqian Jiang, Aili Fan, Yuxin Cui, Yanxing Jia*. Org. Lett. 2011, 13(2), 312–315.
    Download →
    35. “Total Synthesis of Clavicipitic Acid and Aurantioclavine: Stereochemistry of Clavicipitic Acid Revisited”, Zhengren Xu, Weimin Hu, Qiang Liu, Lihe Zhang, Yanxing Jia*. J. Org. Chem. 2010, 75, 7626–7635.
    Download →
    34. “One-Pot AgOAc-Mediated Synthesis of Polysubstituted Pyrroles from Primary Amines and Aldehydes: Application to the Total Synthesis of Purpurone”, Qingjiang Li, Aili Fan, Zhiyao Lu, Yuxin Cui, Wenhan Lin, Yanxing Jia*. Org. Lett. 2010, 12, 4066–4069.
    Download →
    33. “Stereocontrolled and Efficient Total Synthesis of (-)-Stephanotic Acid Methyl Ester and (-)-Celogentin C”, Weimin Hu, Fengying Zhang, Zhengren Xu, Qiang Liu, Yuxin Cui, Yanxing Jia*. Org. Lett. 2010, 12, 956–959.
    Download →
    32. "Water-Controlled Regioselectivity of Pd-Catalyzed Domino Reaction Involving a C–H Activation Process: Rapid Synthesis of Diverse Carbo- and Heterocyclic Skeletons", Zhiyao Lu, Chunmei Hu, Jiajie Guo, Jing Li, Yuxin Cui, Yanxing Jia*. Org. Lett. 2010, 12, 480–483.
    Download →
    31. "Artificial Transcription Factors which Mediate Double-Strand DNA Cleavage", Chao Li, Chao Du, Hua Tian, Chao Jiang, Min Du, Yan Liu, Ren-Zhong Qiao,* Yanxing Jia,* and Yu-Fen Zhao.* Chem. Eur. J. 2010, 16, 12935–12940.
    Download →
    30. “Formal Synthesis of Semiaquilegin A”, Jing Li, Yong Jiang, Qingjiang Li, Qiang Xiao, Yanxing Jia*, Pengfei Tu*. Tetrahedron Lett. 2010, 51, 1121–1123.
    Download →
    29. “Palladium-Catalyzed Synthesis of Tryptamines and Tryptamine Homologues: Synthesis of Psilocin”, Chunmei Hu, Hua Qin, Yuxin Cui, Yanxing Jia*. Tetrahedron 2009, 65, 9075–9080.
    Download →
    28. “Efficient Total Synthesis of (-)-cis-Clavicipitic Acid”, Zhengren Xu, Qingjiang Li, Lihe Zhang, Yanxing Jia*. J. Org. Chem. 2009, 74, 6859–6862.
    Download →
    27. “Total Synthesis of (-)-Incarvilline and (-)-Incarvillateine”, Fengying Zhang, Yanxing Jia*. Tetrahedron 2009, 65, 6840–6843.
    Download →
    26. “Palladium-Catalyzed Indole and Azaindole synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and Chloroaminopyridines with Aldehydes”, Zhengren Xu, Weimin Hu, Fengying Zhang, Qingjiang Li, Zhiyao Lü, Lihe Zhang, Yanxing Jia*. Synthesis 2008, 3981–3987.
    Download →
    Post-doctoral and Ph. D. Work

    25. “Total Synthesis of Complestatin (Chloropeptin II)”, Zhihui Wang, Michèle Bois-Choussy, Yanxing Jia, Jieping Zhu*. Angew. Chem. Int. Ed. 2010, 49, 2018–2022. Angew. Chem. 2010, 122, 2062– 2066.

     

    24. “Synthesis of Diastereomers of Complestatin, and Chloropeptin, High Substrate-dependent Atropstereoselectivity of Intramolecular Suzuki-Miyaura Reaction”, Yanxing Jia, Michèle Bois-Choussy, Jieping Zhu*. Angew. Chem. Int. Ed. 2008, 47, 4167–4172. Angew. Chem. 2008, 120, 4235–4240 .

     

    23. “Synthesis of DEFG Ring of Complestatin and Chloropeptin I: Highly Atropdiastereoselective Macrocyclization by Intramolecular Suzuki-Miyaura Reaction”, Yanxing Jia, Michèle Bois-Choussy, Jieping Zhu*. Org. Lett. 2007, 9, 2401–2404.

     

    22. “Palladium-Catalyzed Enantioselective Domino Heck-Cyanation Sequence: Development and Application to the Total Synthesis of Physostigmine”, Artur Pinto, Yanxing Jia, Luc Neuville, Jieping Zhu*. Chem. -A Eur. J. 2007, 13, 961–967.

     

    21. “Importance of the Structure of Vancomycin Binding Pocket in Designing Compounds Active Against Vancomycin-resistant Enterococci (VRE)”, Yanxing Jia, Michèle Bois-Choussy, Adriano Malabarba, Cristina Brunati, Jieping Zhu*. J. Antibiotics. 2006, 59, 543–552.

     

    20. “Palladium-Catalyzed, Modular Synthesis of Highly Functionalized Indoles and Tryptophans by Direct Annulation of Substituted o-Haloanilines and Aldehydes”, Yanxing Jia, Jieping Zhu*. J. Org. Chem. 2006, 71, 7826–7834.

     

    19. “A Novel Strategy for the Key Fully Substituted Cyclopentenedione Moiety of Madindolines via AlEt3-Promoted Tandem Reductive Rearrangement of a-Hydroxy Epoxides”, Shuanhu Gao, Yanxing Jia, Xuezhi Zhao, Yongqiang Tu*. Chin. J. Chem. 2006, 24, 595– 597.

     

    18. “Design and Synthesis of Simple Macrocycles Active Against    Vancomycin-resistant Enterococci (VRE)”, Yanxing Jia, Nianchun Ma, Zuosheng Liu, Michèle Bois-Choussy, Eduardo Gonzalez-Zamora, Adriano Malabarba, Cristina Brunati, Jieping Zhu*. Chem. Eur. J. 2006, 12, 5334–5351.

     

    17. “Synthesis of Ring-A-Substituted Tryptophan by a Palladium-Catalyzed Heteroannulation Reaction”, Yanxing Jia, Jieping Zhu*. Synlett 2005, 2469–2472.

     

    16. “Identification of Synthetic Compounds Active Against VRE: The Role of the Lipidated Aminoglucose and the Structure of Glycopeptide Binding Pocket”, Yanxing Jia, Eduarda Gonzalez-Zamora, Nianchun Ma, Zuosheng Liu, Michèle Bois-Choussy, Adriano Malabarba, Cristina Brunati, Jieping Zhu*. Bioorg. Med. Chem. Lett. 2005, 15, 4594–4599.

     

    15. “Synthesis of b-Amino-a-Hydroxy Esters and b-Amino-a-Azido Ester by Sharpless Asymmetric Aminohydroxylation, By-Products Analysis”, Zuosheng Liu, Nianchun Ma, Yanxing Jia, Michèle Bois-Choussy, Adriano Malabarba, Jieping Zhu*. J. Org. Chem. 2005, 70, 2847– 2850.

     

    14. “Design and synthesis of macrocycles active against vancomycin-resistant enterococci (VRE): the interplay between D-Ala-D-Lac binding and hydrophobic effect”, Nianchun Ma, Yanxing Jia, Zuosheng Liu, Eduarda Gonzalez-Zamora, Michèle Bois-Choussy, Adriano Malabarba, Cristina Brunati, Jieping Zhu*. Bioorg. Med. Chem. Lett. 2005, 15, 743–746.

     

    13. “Synthetic studies of the HIV-1 protease inhibitive didemnaketals: stereocontrolled synthesis of an ester side chain”, Xuezhi Zhao, Yongqiang Tu,* Lei Peng, Xueqiang Li, Yanxing Jia. Tetrahedron Lett. 2004, 45, 3713–3716.

     

    12. “An Interesting AlEt3-promoted Stereoselective Tandem Rearrangement/ Reduction of a-Hydroxy (or Amino) Heterocyclopropane”, Xin Li, Bin Wu, Xuezhi Zhao, Yanxing Jia, Yongqiang Tu*, Derun Li. Synlett 2003, 623–626.

     

    11. “An efficient synthetic approach to the aromatic sesquiterpenoids via a SmI2-promoted construction of quternary centre”, Xuezhi Zhao, Yanxing Jia, Yongqiang Tu*. J. Chem. Res(S). 2003, 27, 54–55.

     

    10. “Convergent synthesis of the key core spiroketals of the HIV-1 protease inhibitors didemnaketals”, Yanxing Jia, Xin Li, Pingzhen Wang, Bin Wu, Xuezhi Zhao, Yongqiang Tu*. J. Chem. Soc., Perkin trans. 1 2002, 565–570.

     

    9. “A convergent synthesis of the spiroketal moiety of the HIV-1 protease inhibitors didemnaketals”, Yanxing Jia, Xin Li, Bin Wu, Xuezhi Zhao, Yongqiang Tu*. Tetrahedron 2002, 58, 1697–1708.

     

    8. “Synthetic Studies of the HIV-1 Protease Inhibitive Didemnaketals: Stereocontrolled Synthetic Approach to the Key Mother Spiroketals”, Yanxing Jia, Bin Wu, Xin Li, Shikuo Ren, Yongqiang Tu,* Albert S. C. Chan, William Kitching. Org. Lett. 2001, 3, 847–849.

     

    7. “A New One-Pot Synthesis of 2-Quaternary 1,3-Diketones”, Shikuo Ren, Fei Wang, Huani Dou, Chunan Fan, Lan He, Zhenlei Song, Wujiong Xia, Derun Li, Yanxing Jia, Xin Li, Yong qiang Tu*. Synthesis 2001, 16, 2384–2388.

     

    6. “Diastereo-recognizable reaction between Cr(VI) reagents and tertiary a-hydroxy epoxide”, Yongqiang Tu,* Shikuo Ren, Yanxing Jia, Baomin Wang, Albert S. C. Chan, Michael C. K. Choi. Tetrahedron Lett. 2001, 42, 2141–2144.

     

    5. “手性3,7-二甲基-5,6-二羟基-辛-7-烯醛中间体的合成”，贾彦兴, 吴滨, 涂永强*, 高等学校化学学报. 2001, 22, 584-586.

     

    4. “Synthetic Studies of Didemnaketals Analogue-Construction of the Intermediate (3S,5S,6R)-3,7-Dimethyl-5,6,7-trihydroxy-octanal”, Yanxing Jia, Bin Wu, Pingzhen Wang, Yongqiang Tu*. Chin. Chem. Lett. 2000, 11, 509–510.

     

    3. “Didemnaketal A 类似物的合成研究- C1-C7 中间体的合成”，贾彦兴, 王平珍, 吴滨, 涂永强*, 高等学校化学学报. 2000, 21, 729-730.

     

    2. “Synthetic Studies of an Analogue of HIV-1 Protease Inhibitors of Didemnaketals: Constructionof the C1-C8 Intermediate”, Pingzhen Wang, Yanxing Jia, Yongqiang Tu*, Bin Wu. Chin. Chem. Lett. 1999, 10, 749–750.

     

    1. “Didemnaketal A 类似物的合成研究- C8-C15中间体的合成”, 涂永强*, 刘增路, 王平珍, 贾彦兴, 高等学校化学学报. 1999, 20, 81-83.

    专著教材：

    6. 《医用化学》，第17章-含氮有机化合物，贾彦兴，201707；主编：杨峰，孙体健。高等教育出版社

     

    5. “MBFTs for the total synthesis of natural products” in “Stereoselective Multiple Bond-Transformations (MBFTs)”, Eds. Rodriguez, J.; Bonne, D. John Wiley & Sons, Inc 2015, ch13, 365-392. Yanxing Jia,*  Shiqiang Zhou.

     

    4. 《海洋药物导论》，第15章-化学合成研究，贾彦兴，2012年9月；主编：张文。上海科学出版社。

     

    3. 《医用化学》，第18章-有机含氮化合物，贾彦兴，2011；主编：杨峰，孙体健。科学出版社。

     

    2. “One or More C-H Bond(s) Formed by Substitution: Reduction of Carbon-Nitrogen, -Phosphorus, -Arsenic, -Antimony, -Bismuth, -Carbon, -Silicon, -Germanium, -Boron, and –Metal Bonds” in “Comprehensive Organic Functional Group Transformations II”, Eds. Katritzky, A. R., Taylor, R. J. K.; Volume Ed. Cossy, J. Elsevier, 2005, 1, 31-78. Jérome Blanchet, Yanxing Jia, Jieping Zhu*

     

    1. “4-Nitrophenyltriflate” in Electronic Encyclopedia of Reagents for Organic Synthesis (e-EROS) Ed; L. A. Paquette, Wiley-VCH, Weinheim. 2004. Yanxing Jia, Jieping Zhu*

    Patents

    7. 刘海超，贾彦兴；麦角类生物碱的不对称合成方法。申请号： 201710597742.0；申请日：2017-7-20。

     

    6. 杨巧，李磊，贾彦兴；加兰他敏和力克拉敏的不对称合成方法。申请号：201410800466.X；申请日：2014-12-22。授权日：2016-8-24，专利批准号：ZL 201410800466.X。

     

    5. 张丰盈，王斌，黄斌，贾彦兴；角蒿酯碱类似物及其制备方法和在镇痛药物中的应用。申请号：201110254018.0；申请日：2011-8-31。授权日：2016-7-13，专利批准号：ZL 2011 1 0254018.0。

     

    4. 范爱丽，林文翰，贾彦兴，徐岷娟；Baculiferin L及其类似物的制备方法和抗艾滋病用途。申请号：201110077956.8；申请日：2011-3-30。

     

    3. 覃华，贾彦兴；取代吲哚并内酰胺衍生物的制备及作为抗疟疾的用途。

    申请号：201110009088.X；申请日：2011-1-17。

     

    2. 李清江，贾彦兴；1，3，4-三取代或3，4二取代的吡咯环化合物的制备方法。申请号：201010177801.7；申请日：2010-5-14。授权日期：2013-8-7，专利批准号：ZL 2010 1 0177801.7。

     

    1. 姜勇，李菁，贾彦兴，屠鹏飞；一种制备长栲利素A的方法。申请号：200910236592.6; 申请日：2009-11-3。授权日期：2012-9-26，专利批准号：ZL 2009 1 0236592.6。